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| Compound Name: | [9-O-C3H3]-(+)-a-Dihydrotetrabenazine |
| NIMH Code: | D-911 |
| Alternative Name: | |
| Abbreviation: | |
| Indications: | Tritiated analog of the active metabolite of tetrabenazine with high affinity for the vesicular monamine transporter (VMAT2). |
| Package Sizes: | |
| References: | M. R. Kilbourne, L. C. Lee, M. J. Heeg and D. M. Jewett, Absolute configuration of (+)-alpha-dihydrotetrabenazine, an active metabolite of tetrabenazine, Chirality, 9, 59-62 (1997); M. Kilbourne, L. Lee, T. Vander Borght, D. Jewett and K. Frey, Binding of alpha-dihydrotetrabenazine to the vasicular monoamine transporter is stereospecific, Eur. J. Pharmacol., 278, 249-252 (1995). |
| CAS: | |
| Molecular Formula: | C19 H29 N O3 |
| HBA: | 4 |
| HBD: | 1 |
| RotB: | 4 |
| PubChemID: | |
| AlogP: | 3.1 |
| TPSA: | 41.9 |
| Activity: | Dopamine uptake inhibitor (radiolabeled) |
| Comments: | |
| Last Updated 2008-12-09 03:50 PM | |