NIMH Chemical Synthesis and Drug Supply Program

Compound Information Page

Compound Name: [3H]PNU-101,958
NIMH Code: P-901
Alternative Name: [N3H3]-1-Benzyl-4-[N-(3-isopropoxy-2-pyridyl)-N-methyl]aminopiperidine
Package Sizes:
References: R. de la Garza, II and B. K. Madras, [3H]PNU-101958, a D4 dopamine receptor probe, accumulates in prefrontal cortex and hippocampus of non-human primate brain, Synapse, 37, 232-244 (2000); N. S. Kula, F. I. Tarazi, R. J. Baldessarini, L. Xu, V. Bakthavachalam, S. Pounds and C. D. True, Neuropharmacological assessment of potential dopamine D4 receptor-selective radioligands, Eur. J. Pharmacol., 367, 139-142 (1999).
Molecular Formula: C21H26T3N3O
HBA: 4
HBD: 0
RotB: 6
AlogP: 3.9533
TPSA: 28.6
Comments: Specific activity: 85 Ci/mmol
Last Updated 2008-03-04 03:00 PM
Structure of P-901
About The Program

Since 1959, the NIMH Chemical Synthesis and Drug Supply Program has synthesized and distributed novel research chemicals, psychoactive drugs, and compounds that are unavailable from commercial sources to the scientific community working on research relevant to mental health.

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