NIMH Chemical Synthesis and Drug Supply Program

Compound Information Page

Compound Name: Iodine-125 Labeled Epidepride
NIMH Code: E-901
Alternative Name:
Abbreviation:
Indications: picomolar dopamine D2 receptor ligand
Package Sizes:
References: J. A. Clanton, T. de Paulis, D. E. Schmidt, M. S. Ansari, R. G. Manning, R. W. Baldwin and R. M. Kessler, Preparation of [123I] and [125I]epidepride: a dopamine D-2 receptor antagonist radioligand, J. Labelled Comp. Radiopharm., XXIX, 745-751 (1991).
CAS: 107188-87-4
Molecular Formula: C16H23IN2O3
HBA: 4
HBD: 1
RotB: 6
PubChemID: 449726
AlogP: 2.1472
TPSA: 50.8
Activity:
Comments: Most recent batch synthesized 01/30/2006. Shipped in a 73:27 A:B mixture with A being 20 mM sodium hydrogen phosphate/sodium dihydrogen phosphate (pH 6.3) and B being 95% ethanol. Specific activity is 2,175 Ci/mmol. Radiochemical purity is 99%.
Last Updated 2008-11-11 02:43 PM
Structure of E-901
About The Program

Since 1959, the NIMH Chemical Synthesis and Drug Supply Program has synthesized and distributed novel research chemicals, psychoactive drugs, and compounds that are unavailable from commercial sources to the scientific community working on research relevant to mental health.

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