NIMH Chemical Synthesis and Drug Supply Program

Compound Information Page

Compound Name: GBR 12909 Dihydrochloride
NIMH Code: G-801
Alternative Name: 1-[2-[bis(4-Fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine Dihydrochloride
Abbreviation: GBR 12909 Dihydrochloride
Indications: dopamine reuptake inhibitor with behavioral effects similar to cocaine
Package Sizes:
References: K. F. Melia and R. D. Spealman, Pharmacological characterization of the discriminative-stimulus effects of GBR 12909, J. Pharmacol. Exp. Ther., 258, 626-632 (1991); R. E. Heikkila and L. Manzino, Behavioral properties of GBR 12909, GBR 13069 and GBR 13098: specific inhibitors of dopamine uptake, Eur. J. Pharmacol., 103, 241-248 (1984).
CAS: 67469-78-7
Molecular Formula: C28H34Cl2F2N2O
HBA: 5
HBD: 0
RotB: 10
PubChemID: 3455
AlogP: 6.1208
TPSA: 15.71
Activity: Dopamine Uptake Inhibitor
Last Updated 2008-11-11 02:44 PM
Structure of G-801
About The Program

Since 1959, the NIMH Chemical Synthesis and Drug Supply Program has synthesized and distributed novel research chemicals, psychoactive drugs, and compounds that are unavailable from commercial sources to the scientific community working on research relevant to mental health.

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