Compound Information Page
| NIMH Code: | N-905 |
| Compound Name: | (-)-(2S,4R)-1-{(3R)-5-Chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxyphenyl)-2-oxo-2,3-dihydro-1H-indol-3-yl}-4-hydroxy-N,N-dimethyl-2-pyrrolidine-carboxamide |
| Alternative Name: | (2S,4R)-1-[(3R)-5-chloro-1-(2,4-dimethoxyphenyl)sulfonyl-3-(2-methoxyphenyl)-2-oxoindol-3-yl]-4-hydroxy-N,N-dimethylpyrrolidine-2-carboxamide |
| Abbreviation: | Nelivaptan |
| PubChemID: | 9895468 |
| CAS: | 439687-69-1 |
| Molecular Formula: | C30H32ClN3O8S |
| Biological Activity: | Orally-active non-peptide vasopressin V1b receptor antagonist |
| References: | Serradeil-Le Gal, C.; Wagnon, J.; Simiand, J.; Griebel, G.; Lacour, C.; Guillon, G.; Barberis, C.; Brossard, G.; Soubrié, P.; Nisato, D.; Pascal, M.; Pruss, R.; Scatton, B.; Maffrand, J. P.; Le Fur, G. J. Pharmacol. Exp. Ther. 2002, 300, 1122-1130. Serradeil-Le Gal, C.; Wagnon, J.; Tonnerre, B.; Roux, R.; Garcia, G.; Griebel, G.; Aulombard, A. CNS Drug Rev. 2005, 11, 53-68. |
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| Last Updated 2021-03-15 07:46 AM | |
